Etizolam 1 MG Pellets – Thienodiazepine Laboratory Grade Research Formulation

Overview of Etizolam

Etizolam is a thienodiazepine analog with potent anxiolytic, sedative, and muscle-relaxant properties. These 1 mg pellets were developed for controlled studies of GABA-A receptor interactions and neuropharmacological processes. 1V-LSD 150 MCG Blotters

Produktfunktioner

• Exactly 1 mg Etizolam per pellet (±2% variation)
• Formulated with microcrystalline cellulose
• Photostable and moisture-resistant packaging
• Batch checked for:
  • HPLC purity (≥98%)
  • MS Identity Verification
  • Weight and size uniformity

Pharmacological Profile

• High affinity for GABA-A receptors
• Selective binding to α1–α5 subtypes
• Pharmacological action:
  • Anxiolytic
  • Sedative
  • Muscle relaxant
• Shorter elimination half-life than classical benzodiazepines

Application areas in Research

1. Neurofarmakologi
   • GABA-A receptor interactions
   • Allosteric modulation
   • Subtype specificity
2. Comparative Analysis
   • Structure-activity comparison with benzodiazepines
   • Metabolic pathway research
3. Behavioral science
   • Anxiety models (e.g. EPM, OFT)
   • Sleep and wake cycles
   • Convulsion suppression

Tekniske specifikationer

• Pellet diameter: 2.5 mm ± 0.1 mm
• Weight: 10 mg ± 0.5 mg
• Color: Pure white
• Solubility: >5 mg/ml in ethanol (96%)
• Melting point: 146–148°C

Stability profile

• Shelf life: 36 months at 15–25°C
• Light fastness: <1% degradation/year
• Moisture content: <0.5% (Karl Fischer)

Dosage Guidelines (For Reference Only)

• In vitro: 10–1000 nM
• Preclinical: 0.05–0.5 mg/kg
• Behavioral models: 0.1–1.0 mg/kg

Safety and Storage Information

• Store in light-proof packaging
• Relative humidity <40%
• Temperature between 15–25°C
• Compatible with PBS, NaCl 0.9% O-DSMT 50 mg pellets

Dokumentation ved levering

• COA with:
  • Renhed
  • Retention time
  • Mass identification
• Safety Data Sheet (SDS) according to GHS
• Technical sheet with:
  • Stability data
  • Experimental design proposals
  • Solubility analysis

For scientific purposes only. Not suitable for medical, diagnostic, or human consumption. Caluanie Muelear Oxider