{"id":23116,"date":"2025-04-13T17:39:10","date_gmt":"2025-04-13T17:39:10","guid":{"rendered":"https:\/\/researchchemicalhub.com\/?post_type=product&#038;p=23116"},"modified":"2025-10-30T12:49:20","modified_gmt":"2025-10-30T12:49:20","slug":"%d8%ad%d8%a8%d9%8a%d8%a8%d8%a7%d8%aa-%d8%a5%d9%8a%d8%aa%d9%8a%d8%b2%d9%88%d9%84%d8%a7%d9%85-1-%d9%85%d9%84%d8%ba","status":"publish","type":"product","link":"https:\/\/researchchemicalhub.com\/ar\/%d9%85%d8%ad%d9%84\/%d9%85%d9%8f%d8%ad%d8%b1%d9%91%d9%8e%d9%85\/%d8%ad%d8%a8%d9%8a%d8%a8%d8%a7%d8%aa-%d8%a5%d9%8a%d8%aa%d9%8a%d8%b2%d9%88%d9%84%d8%a7%d9%85-1-%d9%85%d9%84%d8%ba\/","title":{"rendered":"\u062d\u0628\u064a\u0628\u0627\u062a \u0625\u064a\u062a\u064a\u0632\u0648\u0644\u0627\u0645 1 \u0645\u0644\u063a"},"content":{"rendered":"<h1><strong><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Etizolam 1 MG Pellets \u2013 Thienodiazepine Laboratory Grade Research Formulation<\/span><\/span><\/strong><\/h1>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Overview of Etizolam<\/span><\/span><\/h2>\n<p><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Etizolam is a thienodiazepine analog with potent anxiolytic, sedative, and muscle-relaxant properties. These 1 mg pellets were developed for controlled studies of GABA-A receptor interactions and neuropharmacological processes. <\/span><\/span><a href=\"https:\/\/researchchemicalhub.com\/ar\/%d9%85%d8%ad%d9%84\/%d9%84%d9%8a%d8%b3%d8%b1%d8%ac%d8%a7%d9%85%d9%8a%d8%af%d8%a7%d8%aa\/1vlsd\/\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">\u0646\u0634\u0627\u0641\u0627\u062a 1V-LSD 150 MCG<\/span><\/span><\/a><\/p>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">\u0645\u0645\u064a\u0632\u0627\u062a \u0627\u0644\u0645\u0646\u062a\u062c<\/span><\/span><\/h2>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Exactly 1 mg Etizolam per pellet (\u00b12% variation)<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Formulated with microcrystalline cellulose<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Photostable and moisture-resistant packaging<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Batch checked for:<\/span><\/span>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">HPLC purity (\u226598%)<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">MS Identity Verification<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Weight and size uniformity<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<\/ul>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Pharmacological Profile<\/span><\/span><\/h2>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">High affinity for GABA-A receptors<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Selective binding to \u03b11\u2013\u03b15 subtypes<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Pharmacological action:<\/span><\/span>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Anxiolytic<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Sedative<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Muscle relaxant<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Shorter elimination half-life than classical benzodiazepines<\/span><\/span><\/li>\n<\/ul>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Application areas in Research<\/span><\/span><\/h2>\n<ol>\n<li><strong><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">\u0639\u0644\u0645 \u0627\u0644\u0623\u062f\u0648\u064a\u0629 \u0627\u0644\u0639\u0635\u0628\u064a\u0629<\/span><\/span><\/strong>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">GABA-A receptor interactions<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Allosteric modulation<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Subtype specificity<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<li><strong><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Comparative Analysis<\/span><\/span><\/strong>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Structure-activity comparison with benzodiazepines<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Metabolic pathway research<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<li><strong><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Behavioral science<\/span><\/span><\/strong>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Anxiety models (e.g. EPM, OFT)<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Sleep and wake cycles<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Convulsion suppression<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<\/ol>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">\u0627\u0644\u0645\u0648\u0627\u0635\u0641\u0627\u062a \u0627\u0644\u0641\u0646\u064a\u0629<\/span><\/span><\/h2>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Pellet diameter: 2.5 mm \u00b1 0.1 mm<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Weight: 10 mg \u00b1 0.5 mg<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">\u0627\u0644\u0644\u0648\u0646: \u0623\u0628\u064a\u0636 \u0646\u0642\u064a<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">\u0627\u0644\u0630\u0648\u0628\u0627\u0646: &gt;5 \u0645\u0644\u063a\/\u0645\u0644 \u0641\u064a \u0627\u0644\u0625\u064a\u062b\u0627\u0646\u0648\u0644 (96%)<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Melting point: 146\u2013148\u00b0C<\/span><\/span><\/li>\n<\/ul>\n<h3><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">\u0645\u0644\u0641 \u0627\u0644\u0627\u0633\u062a\u0642\u0631\u0627\u0631<\/span><\/span><\/h3>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Shelf life: 36 months at 15\u201325\u00b0C<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Light fastness: &lt;1% degradation\/year<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Moisture content: &lt;0.5% (Karl Fischer)<\/span><\/span><\/li>\n<\/ul>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Dosage Guidelines (For Reference Only)<\/span><\/span><\/h2>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">\u0641\u064a \u0627\u0644\u0645\u062e\u062a\u0628\u0631: 10-1000 \u0646\u0627\u0646\u0648\u0645\u0648\u0644<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Preclinical: 0.05\u20130.5 mg\/kg<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Behavioral models: 0.1\u20131.0 mg\/kg<\/span><\/span><\/li>\n<\/ul>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Safety and Storage Information<\/span><\/span><\/h2>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Store in light-proof packaging<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Relative humidity &lt;40%<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Temperature between 15\u201325\u00b0C<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Compatible with PBS, NaCl 0.9% <\/span><\/span><a href=\"https:\/\/researchchemicalhub.com\/ar\/%d9%85%d8%ad%d9%84\/pellets\/%d8%ad%d8%a8%d9%8a%d8%a8%d8%a7%d8%aa-o-dsmt-50mg\/\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">\u062d\u0628\u064a\u0628\u0627\u062a O-DSMT 50 \u0645\u062c\u0645<\/span><\/span><\/a><\/li>\n<\/ul>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">\u0627\u0644\u062a\u0648\u062b\u064a\u0642 \u0639\u0646\u062f \u0627\u0644\u062a\u0633\u0644\u064a\u0645<\/span><\/span><\/h2>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">COA with:<\/span><\/span>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">\u0646\u0642\u0627\u0621<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Retention time<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Mass identification<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Safety Data Sheet (SDS) according to GHS<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Technical sheet with:<\/span><\/span>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">\u0628\u064a\u0627\u0646\u0627\u062a \u0627\u0644\u0627\u0633\u062a\u0642\u0631\u0627\u0631<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Experimental design proposals<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Solubility analysis<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<\/ul>\n<p><em><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">For scientific purposes only. Not suitable for medical, diagnostic, or human consumption. <\/span><\/span><a href=\"https:\/\/researchchemicalhub.com\/ar\/%d9%85%d8%ad%d9%84\/top-10-research-chemicals\/%d8%a3%d9%83%d8%b3%d8%af%d8%a9-%d9%83%d8%a7%d9%84%d9%88%d8%a7%d9%86%d9%8a-%d9%85%d9%8a%d9%88%d9%84%d9%8a%d8%b1\/\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">\u0643\u0627\u0644\u0648\u0627\u0646\u064a \u0645\u0648\u064a\u0644\u064a\u0631 \u0623\u0643\u0633\u062f\u0629<\/span><\/span><\/a><\/em><\/p>","protected":false},"excerpt":{"rendered":"<h2><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Etizolam pellets properties<\/span><\/span><\/span><\/span><\/h2>\n<p><strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Synonym<\/span><\/span><\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"> : 4-(2-chlorophenyl)-2-ethyl-9-methyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine <\/span><\/span><\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">CAS Number<\/span><\/span><\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"> : 40054-69-1 <\/span><\/span><\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Formula<\/span><\/span><\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"> : C17H15ClN4S <\/span><\/span><\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Molar mass<\/span><\/span><\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"> : 342.8 g\/mol <\/span><\/span><\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Purity<\/span><\/span><\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"> : \u2265 99%<\/span><\/span><\/span><\/span><\/p>\n","protected":false},"featured_media":28517,"comment_status":"closed","ping_status":"closed","template":"","meta":[],"product_brand":[82],"product_cat":[488],"product_tag":[917,1130,326],"class_list":{"0":"post-23116","1":"product","2":"type-product","3":"status-publish","4":"has-post-thumbnail","6":"product_brand-research-chemical","7":"product_cat-verboden","8":"product_tag-etizolam","9":"product_tag-etizolam-kopen","10":"product_tag-nl","12":"first","13":"instock","14":"taxable","15":"shipping-taxable","16":"purchasable","17":"product-type-simple"},"_links":{"self":[{"href":"https:\/\/researchchemicalhub.com\/ar\/wp-json\/wp\/v2\/product\/23116","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/researchchemicalhub.com\/ar\/wp-json\/wp\/v2\/product"}],"about":[{"href":"https:\/\/researchchemicalhub.com\/ar\/wp-json\/wp\/v2\/types\/product"}],"replies":[{"embeddable":true,"href":"https:\/\/researchchemicalhub.com\/ar\/wp-json\/wp\/v2\/comments?post=23116"}],"version-history":[{"count":6,"href":"https:\/\/researchchemicalhub.com\/ar\/wp-json\/wp\/v2\/product\/23116\/revisions"}],"predecessor-version":[{"id":28774,"href":"https:\/\/researchchemicalhub.com\/ar\/wp-json\/wp\/v2\/product\/23116\/revisions\/28774"}],"wp:featuredmedia":[{"embeddable":true,"href":"https:\/\/researchchemicalhub.com\/ar\/wp-json\/wp\/v2\/media\/28517"}],"wp:attachment":[{"href":"https:\/\/researchchemicalhub.com\/ar\/wp-json\/wp\/v2\/media?parent=23116"}],"wp:term":[{"taxonomy":"product_brand","embeddable":true,"href":"https:\/\/researchchemicalhub.com\/ar\/wp-json\/wp\/v2\/product_brand?post=23116"},{"taxonomy":"product_cat","embeddable":true,"href":"https:\/\/researchchemicalhub.com\/ar\/wp-json\/wp\/v2\/product_cat?post=23116"},{"taxonomy":"product_tag","embeddable":true,"href":"https:\/\/researchchemicalhub.com\/ar\/wp-json\/wp\/v2\/product_tag?post=23116"}],"curies":[{"name":"\u0648\u0648\u0631\u062f\u0628\u0631\u064a\u0633","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}